Chemical Structure
Antagonist
1650 Citations
Naloxone Hydrochloride
BT-0024
Naloxone is a competitive opioid receptor antagonist used to reverse opioid overdose and as a pharmacological tool in addiction research.
Biological Activity
Competitively blocks μ, κ, and δ opioid receptors, reversing opioid-induced analgesia, sedation, and respiratory depression.
Product Specifications
CAS Number357-08-4
Molecular FormulaC19H22ClNO4
Molecular Weight363.84 g/mol
TargetOpioid Receptor (μ, κ, δ)
PathwayOpioid Receptor Signaling
Disease AreaNeuroscience
IC50/EC50/KdKi: 1.3 nM (μ-OR), 3.5 nM (κ-OR)
Purity>99%
SolubilityWater: ≥50 mg/mL
StorageRoom temperature
SpeciesHuman, Mouse, Rat
Available Sizes
| Size | Price | |
|---|---|---|
| 100 mg | $20.00 | |
| 500 mg | $65.00 |